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Para-Aminosalicylic acid is a prodrug targeting dihydrofolate reductase in Mycobacterium tuberculosis33991
J.Biol.Chem., Volume 288, Issue 32, Number 23456, p.23447- 23456 (2013) Keywords: 0 a acid Activity Agent Agents Aminosalicylic Acid an antagonists & inhibitors Antitubercular Agents article AS Bacterial ...
Ethionamide boosters. 2. Combining bioisosteric replacement and structure-based drug design to solve pharmacokinetic issues in a series of potent 1,2,4-oxadiazole EthR inhibitors31058
Keywords: 0 a Administration,Oral Agent Agents Animals antagonists & inhibitors Antibiotic Antitubercular Agents article Cell Line chemical synthesis chemistry Combination Control Crystallography,X-Ray de ...
Anti-TNF-alpha therapy does not ameliorate disease in a model of acute virus-endotoxin mediated respiratory disease in pigs36852
Keywords: 0 a Activity acute Acute Disease ALL analysis Animal Animals antagonists & inhibitors article AS at Autoimmune Diseases Belgium Bronchoalveolar Lavage Fluid Cell Clinical conditions Control ...
Synthetic EthR inhibitors boost antituberculous activity of ethionamide36849
& inhibitors Antitubercular Agents article AS Binding Sites chemistry concept conventional culture de DNA-Binding Proteins DRUG Drug Resistance Drug Synergism drug therapy drugs effect effects ...
Oseltamivir-resistant influenza virus A (H1N1), Europe, 2007-08 season36834
Source: Emerg.Infect.Dis., Volume 15, Issue 4, Number 560, p.552- 560 (2009) Keywords: 0 2007 2008 a Activity acute Agent Agents antagonists & inhibitors Antiviral Agents article classification Clinical ...
Identification of endomorphin-1 and endomorphin-2 binding sites in human mu-opioid receptor by antisense oligonucleotide strategy4389
Number 512, p.507- 512 (2008) Keywords: 0 a Aequorin ALL Analgesics Analgesics,Opioid analysis Animals antagonists & inhibitors article AS at Base Sequence Binding Sites Calcium Cell cells chemistry ...
Synthesis and biological activity of endomorphin-2 analogs incorporating piperidine-2-, 3- or 4-carboxylic acids instead of proline in position 24391
Number 94, p.91- 94 (2008) Keywords: 0 acid Acids Activity Aequorin Amino Acid Substitution Amino acids an Animals antagonists & inhibitors article AS brain Brain Chemistry Calcium Carboxylic Acids ...
Novel highly potent mu-opioid receptor antagonist based on endomorphin-2 structure4392
Bioorg.Med.Chem.Lett., Volume 18, Issue 4, Number 1353, p.1350- 1353 (2008) Keywords: 0 a Activity Aequorin agonists an Analgesics Analgesics,Opioid Animals antagonists & inhibitors article AS Calcium chemical ...
Mu-opioid receptor ligands lack receptor subtype selectivity in the aequorin luminescence-based calcium assay4393
(2007) Keywords: 0 a Aequorin agonists ALL an analysis Animals antagonists & inhibitors article Calcium Cell cells Change Changes chemistry Cho Cells classification Cricetinae Cricetulus effect ...
Synthesis and characterization of potent and selective mu-opioid receptor antagonists, [Dmt(1), D-2-Nal(4)]endomorphin-1 (Antanal-1) and [Dmt(1), D-2-Nal(4)]endomorphin-2 (Antanal-2)4395
Volume 50, Issue 3, Number 520, p.512- 520 (2007) Keywords: 0 a Aequorin Agent Agents agonists Analgesics Animals antagonists & inhibitors article AS Binding Sites brain Calcium chemical synthesis ...